Ipamorelin — 10 mg
Ipamorelin is a selective pentapeptide GHSR agonist that stimulates pulsatile GH release with minimal ACTH/cortisol activation. Supplied as a 10 mg lyophilised vial for research-only reconstitution. Not for human or veterinary use.
€ 39.00
Description
Ipamorelin 10 mg — Sterling Knight Pharmaceuticals
Category: Peptide / Growth Hormone Secretagogue (GHSR Agonist)
Brand: Sterling Knight Pharmaceuticals
Strength: 10 mg (lyophilised peptide)
Form: Sterile vial for laboratory reconstitution
Packing: 1 × vial
Origin: United Kingdom
Price: €39
Research Use: For qualified laboratory and analytical work only. Not for human or veterinary use.
🧬 What Is Ipamorelin?
Ipamorelin is a synthetic pentapeptide and highly selective agonist of the ghrelin receptor (GHSR1a), designed to stimulate growth hormone (GH) release with minimal effect on ACTH or cortisol. It represents a newer generation of GH secretagogues with improved selectivity compared with classical GHRP peptides.
- Sequence: Aib–His–D-2-Nal–D-Phe–Lys-NH₂
- Class: Growth Hormone Secretagogue (GHSR agonist)
- Molecular Weight: ~711.8 g/mol
- CAS Number: 170851-70-4
Its clean endocrine profile makes it useful for modelling GH pulses and IGF-1 axis behavior without significant adrenal-axis activation.
🔬 Key Research Highlights
1. Selective GHSR Agonism
Ipamorelin activates GHSR1a, inducing pulsatile GH secretion similar to endogenous ghrelin signalling. Importantly, studies show:
- No significant rise in ACTH or cortisol
- Minimal prolactin elevation
- Highly GH-focused endocrine response
2. Human PK/PD Characteristics
- Terminal half-life: ~2 hours
- GH peak occurs at ~0.67 hours post-administration
- Rapid return to baseline, ideal for pulse modelling
3. Anti-Doping Relevance
GHSR agonists and GH-releasing factors, including ipamorelin, are banned by WADA under class S2.
📚 Research Applications
- Modelling GH pulsatility and IGF-1 axis signalling
- Short half-life GH secretagogue for PK/PD experiments
- Reference standard for LC-MS/MS anti-doping method development
- Endocrine pathway studies involving GHSR activation
⚠️ Potential Side Effects & Class-Based Risks
While ipamorelin shows improved selectivity, GH-axis stimulation may cause:
- Headache
- Transient flushing
- Fluid retention / edema
- Alterations in glucose handling (context-dependent)
All GH secretagogues fall under WADA S2, posing doping-test consequences in applicable settings.
Handle strictly as a bioactive peptide with appropriate PPE and biosafety protocols.
🛑 Compliance & Legal Notice
- FOR RESEARCH USE ONLY – Not for human consumption
- Not a medicine, supplement, or veterinary preparation
- Not intended for body enhancement or performance use
- Must be used only by qualified personnel under laboratory SOPs
- WADA Category: S2 — Peptide hormones & releasing factors
📊 Technical Data Table
| Field | Data |
|---|---|
| Chemical Name | Ipamorelin |
| Synonyms | NNC-26-0161; Aib-His-D-2-Nal-D-Phe-Lys-NH₂; Ipamorelin acetate |
| Chemical Formula | C38H49N9O5 |
| Molecular Weight | ≈ 711.8 g/mol |
| CAS Number | 170851-70-4 |
| Total Content | 10 mg lyophilised peptide |
| Stability | 36 months when stored per COA/SDS |
| Origin | United Kingdom |
| Intended Use | Laboratory / analytical / in-vitro research only |
Research chemical — not for human or veterinary use.
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Favorece el crecimiento y la energía de forma natural
Noté mayor resistencia y una recuperación muscular más rápida después de entrenar. Dormí más profundamente y mi energía general estaba más equilibrada. Suave pero efectivo, ideal para quienes buscan un progreso constante.
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Ordine fluido e affidabile
Ho ordinato Ipamorelin 10 mg da CandyGym e ho avuto un’esperienza positiva. La consegna è stata puntuale, l’imballaggio era pulito e il prodotto sembrava autentico. Corrispondeva alla descrizione e offriva un buon rapporto qualità-prezzo.
